BDBM26736 CHEMBL509860::LY2183240::N,N-dimethyl-5-[(4-phenylphenyl)methyl]-1H-1,2,3,4-tetrazole-1-carboxamide
SMILES CN(C)C(=O)n1nnnc1Cc1ccc(cc1)-c1ccccc1
InChI Key InChIKey=GZNIYOXWFCDBBJ-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 26736
Affinity DataIC50: 13nMpH: 7.4 T: 2°CAssay Description:Mouse brain membrane proteomes were preincubated with varying concentrations of inhibitors for 10 min prior to the addition of a rhodamine-tagged flu...More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of mouse brain membrane FAAH preincubated for 10 mins followed by 14C-oleamide substrate addition measured up to 60 mins by TLC analysisMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Louvain Drug Research Institute
Curated by ChEMBL
Louvain Drug Research Institute
Curated by ChEMBL
Affinity DataIC50: 37.3nMAssay Description:Inhibition of human FAAHMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Louvain Drug Research Institute
Curated by ChEMBL
Louvain Drug Research Institute
Curated by ChEMBL
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Louvain Drug Research Institute
Curated by ChEMBL
Louvain Drug Research Institute
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of FAAH (unknown origin)More data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Louvain Drug Research Institute
Curated by ChEMBL
Louvain Drug Research Institute
Curated by ChEMBL
Affinity DataIC50: 38.0nMAssay Description:Inhibition of human recombinant FAAH-maltose binding proteinMore data for this Ligand-Target Pair